P A T E N T

WO2018087347: Use of non-transition metal coordinated dipyridoxyl compounds to prevent and treat chemotherapy-induced PSN

Inventors: Karlsson JOG, Jynge P, Andersson RGG 

PCT filed: 2017

Granted: USA (US10888553B2), Europe (EP3538155B1), China (CN1101396773B), Japan (JP7065866132

Assignee: Karlsson-Tuner Invest AS

Abstract

There is disclosed a platinum ion chelating dipyridoxyl compound, or a pharmaceutically acceptable salt thereof, wherein the dipyridoxyl compound is uncoordinated or coordinated with a metal ion which is not a transition metal, for prevention or treatment of chemotherapy drug induced peripheral sensory neuropathy in a patient, wherein the chemotherapy drug comprises platinum ions. An example of such a chemotherapy drug is oxaliplatin. The drawbacks of previous metal complexed compounds containing manganese ions are eliminated. A more frequent use of the drug is possible since the problem in the prior art with accumulated manganese neurotoxicity is eliminated. The compounds can be administered both temporally and spatially separately from chemotherapy.



WO2013102806A1: Calmangafodipir, a new chemical entity, and other mixed metal complexes, methods of preparation, compositions, and methods of treatment

Inventors: Karlsson JOG, Reineke K, Kurz T, Andersson RGG et al.

PCT filed: 2012

Granted: "Worldwide" 

Assignee: PledPharma AB

Abstract

A mixed metal complex of a compound of Formula I, or a salt thereof, wherein the mixed metals comprise a Group
III-XII transition metal and a Group II metal: (Formula I) (I) wherein X, R 1, R2, R3, and R4 are as defined herein, is produced in a one step crystallization from a solution of the Group III-XII transition metal, the Group II metal, and a compound of Formula I.
Methods for treatment of a pathological condition in a patient, for example, a pathological condition caused by the presence of oxygen-derived free radicals, comprises administering the mixed metal complex to the patient


WO2011004325A1: Pharmaceutical compositions and therapeutic methods employing a combination of a manganese complex compound and a non-manganese complex form of the compound

Inventors: Karlsson JOG, Andersson RGG

PCT filed: 2011

Granted: "Worldvide"

Assignee: PledPharma AB


WO2009078794A1: Compounds for use in the treatment of cancer

Inventors: Karlsson JOG, Kurz T, Andersson RGG

PCT filed: 2007

Granted: "Worldwide"

Assignee: PledPharma AB

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